Tarun Jha

Matrix metalloproteinase-9 (MMP-9) and its inhibitors in cancer: A minireview

European Journal of Medicinal Chemistry · 1970 · journal article

GW170817: Constraining the nuclear matter equation of state from the neutron star tidal deformability

Physical Review C · 1970 · journal article

HDAC6 as privileged target in drug discovery: A perspective

Pharmacological Research · 1970 · journal article

Protease targeted COVID-19 drug discovery and its challenges: Insight into viral main protease (Mpro) and papain-like protease (PLpro) inhibitors

Bioorganic and Medicinal Chemistry · 1970 · journal article

Design of Aminopeptidase N Inhibitors as Anti-cancer Agents

Journal of Medicinal Chemistry · 1970 · journal article

Histone deacetylase 3 (HDAC3) inhibitors as anticancer agents: A review

European Journal of Medicinal Chemistry · 1970 · journal article

Inhibitors of gelatinases (MMP-2 and MMP-9) for the management of hematological malignancies

2021

Chemical-informatics approach to COVID-19 drug discovery: Monte Carlo based QSAR, virtual screening and molecular docking study of some in-house molecules as papain-like protease (PLpro) inhibitors

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Histone deacetylase 8 (HDAC8) and its inhibitors with selectivity to other isoforms: An overview

European Journal of Medicinal Chemistry · 1970 · journal article

Fight against novel coronavirus: A perspective of medicinal chemists

European Journal of Medicinal Chemistry · 1970 · journal article

HDAC3 is a potential validated target for cancer: An overview on the benzamide-based selective HDAC3 inhibitors through comparative SAR/QSAR/QAAR approaches

European Journal of Medicinal Chemistry · 1970 · journal article

Folate decorated epigallocatechin-3-gallate (EGCG) loaded PLGA nanoparticles; in-vitro and in-vivo targeting efficacy against MDA-MB-231 tumor xenograft

International Journal of Pharmaceutics · 1970 · journal article

Combating breast cancer with non-steroidal aromatase inhibitors (NSAIs): Understanding the chemico-biological interactions through comparative SAR/QSAR study

European Journal of Medicinal Chemistry · 1970 · journal article

Is dual inhibition of metalloenzymes HDAC-8 and MMP-2 a potential pharmacological target to combat hematological malignancies?

Pharmacological Research · 1970 · journal article

Design of dual MMP-2/HDAC-8 inhibitors by pharmacophore mapping, molecular docking, synthesis and biological activity

RSC Advances · 1970 · journal article

Chemical-informatics approach to COVID-19 drug discovery: Exploration of important fragments and data mining based prediction of some hits from natural origins as main protease (Mpro) inhibitors

Journal of Molecular Structure · 1970 · journal article

Arylsulfonamides and selectivity of matrix metalloproteinase-2: An overview

European Journal of Medicinal Chemistry · 1970 · journal article

Dissecting Histone Deacetylase 3 in Multiple Disease Conditions: Selective Inhibition as a Promising Therapeutic Strategy

2021

Design, synthesis and biological screening of 2-aminobenzamides as selective HDAC3 inhibitors with promising anticancer effects

European Journal of Pharmaceutical Sciences · 1970 · journal article

Small molecule drug conjugates (SMDCs): an emerging strategy for anticancer drug design and discovery

2021

Exploring pyrazolo[3,4-d]pyrimidine phosphodiesterase 1 (PDE1) inhibitors: a predictive approach combining comparative validated multiple molecular modelling techniques

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Robust design of some selective matrix metalloproteinase-2 inhibitors over matrix metalloproteinase-9 through in silico/fragment-based lead identification and de novo lead modification: Syntheses and biological assays

Bioorganic and Medicinal Chemistry · 1970 · journal article

Selective HDAC3 Inhibitors with Potent In Vivo Antitumor Efficacy against Triple-Negative Breast Cancer

2023

First structure–activity relationship analysis of SARS-CoV-2 virus main protease (Mpro) inhibitors: an endeavor on COVID-19 drug discovery

Molecular Diversity · 1970 · journal article

Assessing structural insights into in-house arylsulfonyl L-(+) glutamine MMP-2 inhibitors as promising anticancer agents through structure-based computational modelling approaches

2023

First molecular modeling report on novel arylpyrimidine kynurenine monooxygenase inhibitors through multi-QSAR analysis against Huntington's disease: A proposal to chemists!

Bioorganic and Medicinal Chemistry Letters · 1970 · journal article

An assessment of crucial structural contributors of HDAC6 inhibitors through fragment-based non-linear pattern recognition and molecular dynamics simulation approaches

2024

5-N-Substituted-2-(substituted benzenesulphonyl) glutamines as antitumor agents. Part II: Synthesis, biological activity and QSAR study

Bioorganic and Medicinal Chemistry · 1970 · journal article

Dual activity of amphiphilic Zn(II) nitroporphyrin derivatives as HIV-1 entry inhibitors and in cancer photodynamic therapy

European Journal of Medicinal Chemistry · 1970 · journal article

Selective inhibition of histone deacetylase 3 by novel hydrazide based small molecules as therapeutic intervention for the treatment of cancer

2022

Studies on the production and purification of an antimicrobial compound and taxonomy of the producer isolated from the marine environment of the Sundarbans

Applied Microbiology and Biotechnology · 1970 · journal article

Design, synthesis, biological evaluation and molecular docking study of arylcarboxamido piperidine and piperazine-based hydroxamates as potential HDAC8 inhibitors with promising anticancer activity

European Journal of Pharmaceutical Sciences · 1970 · journal article

Structure-activity relationships of HDAC8 inhibitors: Non-hydroxamates as anticancer agents

Pharmacological Research · 1970 · journal article

First report on the structural exploration and prediction of new BPTES analogs as glutaminase inhibitors

Journal of Molecular Structure · 1970 · journal article

QSAR study on some pyridoacridine ascididemin analogues as anti-tumor agents

Bioorganic and Medicinal Chemistry · 1970 · journal article

Good and bad molecular fingerprints for human rhinovirus 3C protease inhibition: identification, validation, and application in designing of new inhibitors through Monte Carlo-based QSAR study

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Histone deacetylase 3 inhibitors in learning and memory processes with special emphasis on benzamides

European Journal of Medicinal Chemistry · 1970 · journal article

A new bisbenzylisoquinoline alkaloid isolated from Thalictrum foliolosum, as a potent inhibitor of DNA topoisomerase IB of Leishmania donovani

Fitoterapia · 1970 · journal article

Structure-activity relationships of hydroxamate-based histone deacetylase-8 inhibitors: Reality behind anticancer drug discovery

Future Medicinal Chemistry · 1970 · journal article

Glycyrrhizin as a promising kryptonite against SARS-CoV-2: Clinical, experimental, and theoretical evidences

2022

Synthesis, screening and quantitative structure-activity relationship (QSAR) studies of some glutamine analogues for possible anticancer activity

Bioorganic and Medicinal Chemistry · 1970 · journal article

Tides in merging neutron stars: Consistency of the GW170817 event with experimental data on finite nuclei

Physical Review C · 1970 · journal article

Exploring structural requirements of aurone derivatives as antimalarials by validated DFT-based QSAR, HQSAR, and COMFA-COMSIA approach

Medicinal Chemistry Research · 1970 · journal article

QSAR study on some anti-HIV HEPT analogues using physicochemical and topological parameters

Bioorganic and Medicinal Chemistry · 1970 · journal article

Synergistic effect of methanol extract of Abies webbiana leaves on sleeping time induced by standard sedatives in mice and anti-inflammatory activity of extracts in rats

Journal of Ethnopharmacology · 1970 · journal article

Chrysin-loaded PLGA attenuates OVA-induced allergic asthma by modulating TLR/NF-κB/NLRP3 axis

Nanomedicine: Nanotechnology, Biology, and Medicine · 1970 · journal article

Anthocephaline, a New Indole Alkaloid and Cadambine, a Potent Inhibitor of DNA Topoisomerase IB of <i>Leishmania donovani</i> (LdTOP1LS), Isolated from <i>Anthocephalus cadamba</i>

2015

QSAR study on some p-arylthio cinnamides as antagonists of biochemical ICAM-1/LFA-1 interaction and ICAM-1/JY-8 cell adhesion in relation to anti-inflammatory activity

Bioorganic and Medicinal Chemistry · 1970 · journal article

Synthesis, biological evaluation, and molecular docking analysis of novel linker-less benzamide based potent and selective HDAC3 inhibitors

2021

Cytotoxic potential of dispirooxindolo/acenaphthoquino andrographolide derivatives against MCF-7 cell line

MedChemComm · 1970 · journal article

QSAR study on adenosine kinase inhibition of pyrrolo[2,3-d]pyrimidine nucleoside analogues using the Hansch approach

Bioorganic and Medicinal Chemistry Letters · 1970 · journal article

Hydroxyethylamine derivatives as HIV-1 protease inhibitors: a predictive QSAR modelling study based on Monte Carlo optimization

SAR and QSAR in Environmental Research · 1970 · journal article

Exploring QSAR and pharmacophore mapping of structurally diverse selective matrix metalloproteinase-2 inhibitors

Journal of Pharmacy and Pharmacology · 1970 · journal article

Design of 5-fluorouracil (5-FU) loaded, folate conjugated peptide linked nanoparticles, a potential new drug carrier for selective targeting of tumor cells

MedChemComm · 1970 · journal article

A review on camptothecin analogs with promising cytotoxic profile

Anti-Cancer Agents in Medicinal Chemistry · 1970 · journal article

Diverse classes of HDAC8 inhibitors: In search of molecular fingerprints that regulate activity

Future Medicinal Chemistry · 1970 · journal article

A pentanoic acid derivative targeting matrix metalloproteinase-2 (MMP-2) induces apoptosis in a chronic myeloid leukemia cell line

European Journal of Medicinal Chemistry · 1970 · journal article

Updated chemical scaffolds of ABCG2 inhibitors and their structure-inhibition relationships for future development

2022

Protease targeted COVID-19 drug discovery: What we have learned from the past SARS-CoV inhibitors?

2021

Design, synthesis and binding mode of interaction of novel small molecule o-hydroxy benzamides as HDAC3-selective inhibitors with promising antitumor effects in 4T1-Luc breast cancer xenograft model

2021

Exploring QSAR on 3-aminopyrazoles as antitumor agents for their inhibitory activity of CDK2/cyclin A

European Journal of Medicinal Chemistry · 1970 · journal article

Hot nuclear matter in asymmetry chiral sigma model

Nuclear Physics A · 1970 · journal article

In silico modelling, identification of crucial molecular fingerprints, and prediction of new possible substrates of human organic cationic transporters 1 and 2

New Journal of Chemistry · 1970 · journal article

Insight into the structural requirements of pyrimidine-based phosphodiesterase 10A (PDE10A) inhibitors by multiple validated 3D QSAR approaches

SAR and QSAR in Environmental Research · 1970 · journal article

Are inhibitors of histone deacetylase 8 (HDAC8) effective in hematological cancers especially acute myeloid leukemia (AML) and acute lymphoblastic leukemia (ALL)?

2023

Selective Inhibitors of Medium-Size S1′ Pocket Matrix Metalloproteinases: A Stepping Stone of Future Drug Discovery

2022

Structural findings of phenylindoles as cytotoxic antimitotic agents in human breast cancer cell lines through multiple validated QSAR studies

Toxicology in Vitro · 1970 · journal article

Outline of gelatinase inhibitors as anti-cancer agents: A patent mini-review for 2010-present

European Journal of Medicinal Chemistry · 1970 · journal article

Designing potential HDAC3 inhibitors to improve memory and learning

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Selective and nonselective HDAC8 inhibitors: a therapeutic patent review

Pharmaceutical patent analyst · 1970 · journal article

Comparative validated molecular modeling of p53-HDM2 inhibitors as antiproliferative agents

European Journal of Medicinal Chemistry · 1970 · journal article

Monte Carlo based modelling approach for designing and predicting cytotoxicity of 2-phenylindole derivatives against breast cancer cell line MCF7

Toxicology in Vitro · 1970 · journal article

Quantitative structural assessments of potential meprin β inhibitors by non-linear QSAR approaches and validation by binding mode of interaction analysis

2023

Attributes of a rotating neutron star with a hyperon core

Physical Review C - Nuclear Physics · 1970 · journal article

Antibacterial activity of Abies webbiana

Fitoterapia · 1970 · journal article

A review of MMP-2 structures and binding mode analysis of its inhibitors to strategize structure-based drug design

2022

QSAR study on the affinity of some arylpiperazines towards the 5-HT <inf>1A</inf>/α<inf>1</inf>-adrenergic receptor using the E-state index

Bioorganic and Medicinal Chemistry Letters · 1970 · journal article

Development of decision trees to discriminate HDAC8 inhibitors and non-inhibitors using recursive partitioning

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Understanding Chemico-Biological Interactions of Glutamate MMP-2 Inhibitors through Rigorous Alignment-Dependent 3D-QSAR Analyses

ChemistrySelect · 1970 · journal article

Density functional theory (DFT) studies in HDAC-based chemotherapeutics: Current findings, case studies and future perspectives

2024

Exploring sodium glucose cotransporter (SGLT2) inhibitors with machine learning approach: A novel hope in anti-diabetes drug discovery

2021

Ligand-based Design of Anticancer MMP2 Inhibitors: a Review

2021

Stepwise development of structure-activity relationship of diverse PARP-1 inhibitors through comparative and validated in silico modeling techniques and molecular dynamics simulation

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Structural findings of quinolone carboxylic acids in cytotoxic, antiviral, and anti-HIV-1 integrase activity through validated comparative molecular modeling studies

Medicinal Chemistry Research · 1970 · journal article

Synthesis, pharmacological activity and comparative QSAR modeling of 1,5-N,N′-substituted-2-(substituted naphthalenesulphonyl) glutamamides as possible anticancer agents

European Journal of Medicinal Chemistry · 1970 · journal article

Effective anti-aromatase therapy to battle against estrogen-mediated breast cancer: Comparative SAR/QSAR assessment on steroidal aromatase inhibitors

European Journal of Medicinal Chemistry · 1970 · journal article

Recent trends in fragment-based anticancer drug design strategies against different targets: A mini-review

2022

Bulk viscosity in a hyperonic star and r-mode instability

Physical Review C - Nuclear Physics · 1970 · journal article

Comparative QSAR modelling of 2-phenylindole-3-carbaldehyde derivatives as potential antimitotic agents

Bioorganic and Medicinal Chemistry Letters · 1970 · journal article

Constraints on nuclear matter parameters of an effective chiral model

Physical Review C - Nuclear Physics · 1970 · journal article

Insight into structural features of phenyltetrazole derivatives as ABCG2 inhibitors for the treatment of multidrug resistance in cancer

SAR and QSAR in Environmental Research · 1970 · journal article

Validated predictive QSAR modeling of N-aryl-oxazolidinone-5-carboxamides for anti-HIV protease activity

Bioorganic and Medicinal Chemistry Letters · 1970 · journal article

Structural exploration of hydroxyethylamines as HIV-1 protease inhibitors: new features identified

SAR and QSAR in Environmental Research · 1970 · journal article

Exploring structural requirements of 1-N-substituted thiocarbamoyl-3-phenyl-2-pyrazolines as antiamoebic agents using comparative QSAR modelling

Bioorganic and Medicinal Chemistry Letters · 1970 · journal article

meso-Thiophenium Porphyrins and Their Zn(II) Complexes: A New Category of Cationic Photosensitizers

ACS Medicinal Chemistry Letters · 1970 · journal article

Structural exploration for the refinement of anticancer matrix metalloproteinase-2 inhibitor designing approaches through robust validated multi-QSARs

Journal of Molecular Structure · 1970 · journal article

Possible binding mode analysis of pyrazolo-Triazole hybrids as potential anticancer agents through validated molecular docking and 3D-QSAR modeling approaches

Letters in Drug Design and Discovery · 1970 · journal article

Exploring structural requirements of unconventional Knoevenagel-type indole derivatives as anticancer agents through comparative QSAR modeling approaches

Canadian Journal of Chemistry · 1970 · journal article

Synthesis, biological assessment, and in silico binding mode interaction analyses and DFT studies of biphenylsulfonamide-based potent MMP-2 inhibitors effective against chronic myeloid leukemia

2024

Ligand-based quantitative structural assessments of SARS-CoV-2 3CLpro inhibitors: An analysis in light of structure-based multi-molecular modeling evidences

2021

Molecular dynamics analysis of phytochemicals from Ageratina adenophora against COVID-19 main protease (Mpro) and human angiotensin-converting enzyme 2 (ACE2)

2021

A New Ellagic Acid Glycoside and DNA Topoisomerase IB Inhibitory Activity of Saponins from <i>Putranjiva roxburghii</i>

2014

Leishmanial sphingolipid induces apoptosis in Sarcoma 180 cancer cells through regulation of tumour growth via angiogenic switchover

Tumor Biology · 1970 · journal article

Predictive comparative QSAR modelling of (phenylpiperazinyl-alkyl) oxindoles as selective 5-HT<inf>1A</inf> antagonists by stepwise regression, PCRA, FA-MLR and PLS techniques

European Journal of Medicinal Chemistry · 1970 · journal article

Neutron star matter in an effective model

Physical Review C - Nuclear Physics · 1970 · journal article

QSAR modeling on dopamine D<inf>2</inf> receptor binding affinity of 6-methoxy benzamides

Farmaco · 1970 · journal article

Antitussive activity of Abies webbiana Lindl. Leaf extract against sulphur dioxide-induced cough reflex in mice

Phytotherapy Research · 1970 · journal article

Benzamide porphyrins with directly conjugated and distal pyridyl or pyridinium groups substituted to the porphyrin macrocycles: Study of the photosensitising abilities as inducers of apoptosis in cancer cells under photodynamic conditions

Journal of Photochemistry and Photobiology B: Biology · 1970 · journal article

Pinpointing prime structural attributes of potential MMP-2 inhibitors comprising alkyl/arylsulfonyl pyrrolidine scaffold: a ligand-based molecular modelling approach validated by molecular dynamics simulation analysis

2024

Hyperon bulk viscosity and <i>r</i>-modes of neutron stars

2022

Leishmanial lipid affords protection against oxidative stress induced hepatic injury by regulating inflammatory mediators and confining apoptosis progress

Toxicology Letters · 1970 · journal article

Spermicidal and contraceptive potential of desgalactotigonin: A prospective alternative of nonoxynol-9

PLoS ONE · 1970 · journal article

Exploration of structural and physicochemical requirements and search of virtual hits for aminopeptidase N inhibitors

Molecular Diversity · 1970 · journal article

Quantitative structure-activity relationship study on some benzodiazepine derivatives as anti-Alzheimer agents

Journal of Molecular Modeling · 1970 · journal article

Structural exploration of tetrahydroisoquinoline derivatives as HDAC8 inhibitors through multi-QSAR modeling study

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Reliable structural information for rational design of benzoxazole type potential cholesteryl ester transfer protein (CETP) inhibitors through multiple validated modeling techniques

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Synthesis, anticancer activity, structure-activity relationship and binding mode of interaction studies of substituted pentanoic acids

Future Medicinal Chemistry · 1970 · journal article

Insight into the structural requirements of theophylline-based aldehyde dehydrogenase 1A1 (ALDH1A1) inhibitors through multi-QSAR modeling and molecular docking approaches

Current Drug Discovery Technologies · 1970 · journal article

How the structural properties of the indole derivatives are important in kinase targeted drug design?: A case study on tyrosine kinase inhibitors

2021

Urea transporter and its specific and nonspecific inhibitors: State of the art and pharmacological perspective

2021

Multiple molecular modelling studies on some derivatives and analogues of glutamic acid as matrix metalloproteinase-2 inhibitors^$

SAR and QSAR in Environmental Research · 1970 · journal article

Chenopodium album metabolites act as dual topoisomerase inhibitors and induce apoptosis in the MCF7 cell line

MedChemComm · 1970 · journal article

An updated patent review of matrix metalloproteinase (MMP) inhibitors (2021-present)

2023

Insight into the structural requirement of aryl sulphonamide based gelatinases (MMP-2 and MMP-9) inhibitors – Part I: 2D-QSAR, 3D-QSAR topomer CoMFA and Naïve Bayes studies – First report of 3D-QSAR Topomer CoMFA analysis for MMP-9 inhibitors and jointly inhibitors of gelatinases together

2021

Robust classification-based molecular modelling of diverse chemical entities as potential SARS-CoV-2 3CL^pro inhibitors: theoretical justification in light of experimental evidences

2021

Quantitative activity–activity relationship (QAAR) driven design to develop hydroxamate derivatives of pentanoic acids as selective HDAC8 inhibitors: synthesis, biological evaluation and binding mode of interaction studies

2021

Quantitative Structure-Activity Relationship Study on Some Azidopyridinyl Neonicotinoid Insecticides for Their Selective Affinity Towards the Drosophila Nicotinic Receptor Over Mammalian a4ß2 Receptor Using Electrotopological State Atom Index

2003

Exploring in house glutamate inhibitors of matrix metalloproteinase-2 through validated robust chemico-biological quantitative approaches

Structural Chemistry · 1970 · journal article

Towards the Development of Anticancer Drugs from Andrographolide: Semisynthesis, Bioevaluation, QSAR Analysis and Pharmacokinetic Studies

2015

Lipid from infective L. Donovani regulates acute myeloid cell growth via mitochondria dependent MAPK pathway

PLoS ONE · 1970 · journal article

Quantitative structure-activity relationship study using refractotopological state atom index on some neonicotinoid insecticides

Bioorganic and Medicinal Chemistry · 1970 · journal article

Designing potential antitrypanosomal thiazol-2-ethylamines through predictive regression based and classification based QSAR analyses

Current Drug Discovery Technologies · 1970 · journal article

Identification of structural fingerprints for ABCG2 inhibition by using Monte Carlo optimization, Bayesian classification, and structural and physicochemical interpretation (SPCI) analysis

SAR and QSAR in Environmental Research · 1970 · journal article

An Equation of State for Magnetized Neutron Star Matter and Tidal Deformation in Neutron Star Mergers

Astrophysical Journal · 1970 · journal article

Corrigendum to “Matrix metalloproteinase-9 (MMP-9) and its inhibitors in cancer: A minireview” [Eur. J. Med. Chem. 194 (2020) 112260] (European Journal of Medicinal Chemistry (2020) 194, (S0223523420302270), (10.1016/j.ejmech.2020.112260))

European Journal of Medicinal Chemistry · 1970 · journal article

Exploration of histone deacetylase 8 inhibitors through classification QSAR study: Part II

Journal of Molecular Structure · 1970 · journal article

QSAR modelling on a series of arylsulfonamide-based hydroxamates as potent MMP-2 inhibitors

SAR and QSAR in Environmental Research · 1970 · journal article

Structural refinement and prediction of potential CCR2 antagonists through validated multi-QSAR modeling studies

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Structural insight into the viral 3C-like protease inhibitors: Comparative SAR/QSAR approaches

Viral Proteases and Their Inhibitors · 1970 · book chapter

A combined ligand-based and structure-based <i>in silico</i> molecular modeling approach to pinpoint the key structural attributes of hydroxamate derivatives as promising meprin β inhibitors

2024

Exploring naphthyl derivatives as SARS-CoV papain-like protease (PLpro) inhibitors and its implications in COVID-19 drug discovery

2021

Structural findings of cinnolines as anti-schizophrenic PDE10A inhibitors through comparative chemometric modeling

Molecular Diversity · 1970 · journal article

An overview of matrix metalloproteinase-12 in multiple disease conditions, potential selective inhibitors, and drug designing strategies

2024

Biphenylsulfonamides as effective MMP‐2 inhibitors with promising antileukemic efficacy: Synthesis, in vitro biological evaluation, molecular docking, and MD simulation analysis

2024

A patent review of histone deacetylase 8 (HDAC8) inhibitors (2013–present)

2024

Derivatives of D(−) glutamine-based MMP-2 inhibitors as an effective remedy for the management of chronic myeloid leukemia-Part-I: Synthesis, biological screening and in silico binding interaction analysis

2024

The first report on predictive comparative ligand-based multi-QSAR modeling analysis of 4-pyrimidinone and 2-pyridinone based APJ inhibitors

2022

Quantitative structure activity relationship (QSAR) studies of some substituted benzenesulphonyl glutamines as tumour suppressors.

2001

Leishmanial lipid suppresses the bacterial endotoxin-induced inflammatory response with attenuation of tissue injury in sepsis

Journal of Leukocyte Biology · 1970 · journal article

QSAR modeling of neonicotinoid insecticides for their selective affinity towards Drosophila nicotinic receptors over mammalian α<inf>4</inf>β <inf>2</inf> receptors

Canadian Journal of Chemistry · 1970 · journal article

Exploration of good and bad structural fingerprints for inhibition of indoleamine-2,3-dioxygenase enzyme in cancer immunotherapy using Monte Carlo optimization and Bayesian classification QSAR modeling

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Structural exploration of arylsulfonamide-based ADAM17 inhibitors through validated comparative multi-QSAR modelling studies

Journal of Molecular Structure · 1970 · journal article

Homoisoflavonoids as potential antiangiogenic agents for retinal neovascularization

Biomedicine and Pharmacotherapy · 1970 · journal article

Nuclear symmetry energy with mesonic cross-couplings in the effective chiral model

Physical Review C · 1970 · journal article

Histone deacetylase 8 in focus: Decoding structural prerequisites for innovative epigenetic intervention beyond hydroxamates

2024

Unraveling HDAC11: Epigenetic orchestra in different diseases and structural insights for inhibitor design

2024

Matrix metalloproteinase-8 (MMP-8) and its inhibitors: A minireview

2024

Fragment-based structural exploration and chemico-biological interaction study of HDAC3 inhibitors through non-linear pattern recognition, chemical space, and binding mode of interaction analysis

2023

Binary quantitative activity-activity relationship (QAAR) studies to explore selective HDAC8 inhibitors: In light of mathematical models, DFT-based calculation and molecular dynamic simulation studies

2022

Applying comparative molecular modelling techniques on diverse hydroxamate-based HDAC2 inhibitors: an attempt to identify promising structural features for potent HDAC2 inhibition

2022

Shape change in Hf, W and Os-isotopes: A non-relativistic Hartree-Fock versus relativistic Hartree approximation

2004

A relativistic mean-field study of magic numbers in light nuclei from neutron to proton drip-lines

2003

Ligand based validated comparative chemometric modeling and pharmacophore mapping of aurone derivatives as antimalarial agents

Current Computer-Aided Drug Design · 1970 · journal article

Structural findings of 2-Phenylindole-3-carbaldehyde derivatives for antimitotic activity by FA-sMLR QSAR analysis

Chemical Biology and Drug Design · 1970 · journal article

Essential elements regulating HDAC8 inhibition: a classification based structural analysis and enzyme-inhibitor interaction study of hydroxamate based HDAC8 inhibitors

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

Integrating regression and classification-based QSARs with molecular docking analyses to explore the structure-antiaromatase activity relationships of letrozole-based analogs

Canadian Journal of Chemistry · 1970 · journal article

Exploring the key structural attributes and chemico-biological interactions of pyridinone-based SARS-CoV-2 3CLpro inhibitors through validated structure-based drug design strategies

2024

Fragment-based investigation of thiourea derivatives as VEGFR-2 inhibitors: a cross-validated approach of ligand-based and structure-based molecular modeling studies

2023

Chemometric modeling and pharmacophore mapping in coronary heart disease: 2-arylbenzoxazoles as cholesteryl ester transfer protein inhibitors

MedChemComm · 1970 · journal article

Erratum: Neutron star matter in an effective model (Phys. Rev. C (2006) 74 (055803))

Physical Review C - Nuclear Physics · 1970 · journal article

Evaluation of efficacy of curcumin along with lycopene and piperine in the management of oral submucous fibrosis

Contemporary Clinical Dentistry · 1970 · journal article

An integrated ligand-based modelling approach to explore the structure-property relationships of influenza endonuclease inhibitors

Structural Chemistry · 1970 · journal article

Antineoplastic impact of leishmanial sphingolipid in tumour growth with regulation of angiogenic event and inflammatory response

Apoptosis · 1970 · journal article

Advances in structure-activity relationships of HDAC inhibitors as HIV latency-reversing agents

2024

A fragment-based structural analysis of MMP-2 inhibitors in search of meaningful structural fragments

2022

First molecular modelling report on tri-substituted pyrazolines as phosphodiesterase 5 (PDE5) inhibitors through classical and machine learning based multi-QSAR analysis

2021

Synthesis, biological activity, structure activity relationship study and liposomal formulation development of some arylsulfonyl pyroglutamic acid derivatives

2021

The role of 3D pharmacophore mapping based virtual screening for identification of novel anticancer agents: An overview

Current Topics in Medicinal Chemistry · 1970 · journal article

Possible anticancer agents: QSAR analogs of glutamamide: Synthesis and pharmacological activity of 1,5-N,N′-disubstituted-2-(substituted benzenesulphonyl) glutamamides

European Journal of Medicinal Chemistry · 1970 · journal article

QSAR modelling of pancreatic β-cell K<inf>ATP</inf> channel openers R/S-3,4-dihydro-2,2-dimethyl-6-halo-4-(substituted phenylaminocarbonylamino)-2H-1-benzopyrans using MLR-FA techniques

European Journal of Medicinal Chemistry · 1970 · journal article

Chemometric modeling of 5-Phenylthiophenecarboxylic acid derivatives as anti-rheumatic agents

Current Computer-Aided Drug Design · 1970 · journal article

Cancer photocytotoxicity and anti-inflammatory response ofcis-A<inf>2</inf>B<inf>2</inf>typemeso-p-nitrophenyl andp-hydroxyphenyl porphyrin and its zinc(ii) complex: a synthetic alternative to theTHPPsynthon

New Journal of Chemistry · 1970 · journal article

An integrated QSAR modeling approach to explore the structure–property and selectivity relationships of N-benzoyl-l-biphenylalanines as integrin antagonists

Molecular Diversity · 1970 · journal article

A comparative quantitative structural assessment of benzothiazine-derived HDAC8 inhibitors by predictive ligand-based drug designing approaches

2022

A detail survey and analysis of selectivity criteria for indole-based histone deacetylase 8 (HDAC8) inhibitors

2022

Synthesis, Anticancer Activity, SAR and Binding Mode of Interaction Studies of Substituted Pentanoic Acids: Part II

2021

A robust classification-dependent multi-molecular modelling study on some biphenyl sulphonamide based MMP-8 inhibitors

2021

Enhanced regression of tumors in mice with combined chemotherapy and immunotherapy

2002

Lipid isolated from a Leishmania donovani strain reduces Escherichia coli induced sepsis in mice through inhibition of inflammatory responses

Mediators of Inflammation · 1970 · journal article

Identification of molecular fingerprints of phenylindole derivatives as cytotoxic agents: a multi-QSAR approach

Structural Chemistry · 1970 · journal article

Structural analysis of arylsulfonamide-based carboxylic acid derivatives: a QSAR study to identify the structural contributors toward their MMP-9 inhibition

Structural Chemistry · 1970 · journal article

Unveiling critical structural features for effective HDAC8 inhibition: a comprehensive study using quantitative read-across structure–activity relationship (q-RASAR) and pharmacophore modeling

2024

Modeling Inhibitors of Matrix Metalloproteinases

2023

Employing comparative QSAR techniques for the recognition of dibenzofuran and dibenzothiophene derivatives toward MMP-12 inhibition

2023

Hydrazides as Potential HDAC Inhibitors: Structure-activityRelationships and Biological Implications

2023

Exploration of structural alerts and fingerprints for novel anticancer therapeutics: a robust classification-QSAR dependent structural analysis of drug-like MMP-9 inhibitors

2023

A quantitative structural analysis of AR-42 derivatives as HDAC1 inhibitors for the identification of promising structural contributors

2022

Unmasking of crucial structural fragments for coronavirus protease inhibitors and its implications in COVID-19 drug discovery

2021

Possible antineoplastic agents: Part XIII. Synthesis, biological evaluation and QSAR studies of some 1-(substituted benzenesulphonyl)-5-oxopyrrolidine-2-carboxylic acid derivatives.

1993

Ligand-and structure-based drug design of non-steroidal aromatase inhibitors (NSAIs) in breast cancer

Quantitative Structure-Activity Relationships in Drug Design, Predictive Toxicology, and Risk Assessment · 1970 · book

Collagenases and gelatinases and their inhibitors as anticancer agents

Cancer-Leading Proteases: Structures, Functions, and Inhibition · 1970 · book chapter

Exploring indole derivatives as myeloid cell leukaemia-1 (Mcl-1) inhibitors with multi-QSAR approach: A novel hope in anti-cancer drug discovery

New Journal of Chemistry · 1970 · journal article

Intermolecular association of some selected melanin monomers and their optical absorption

Computational and Theoretical Chemistry · 1970 · journal article

An integrated multi-QSAR modeling approach for designing knoevenagel-type indoles with enhancing cytotoxic profiles

Current Computer-Aided Drug Design · 1970 · journal article

Derivatives of D(−)-glutamine-based MMP-2 inhibitors as an effective remedy for the management of chronic myeloid leukemia-Part-III: Synthesis, biological screening and in silico binding interaction analysis

2024

Antitumor Activity and Antioxidant Role of Ichnocarpus frutescens Against Ehrlich Ascites Carcinoma in Swiss Albino Mice

2007

Exploring the structural aspects of ureido-amino acid-based APN inhibitors: a validated comparative multi-QSAR modelling study

SAR and QSAR in Environmental Research · 1970 · journal article

Shedding light on designing potential meprin β inhibitors through ligand-based robust validated computational approaches: A proposal to chemists!

Journal of Biomolecular Structure and Dynamics · 1970 · journal article

A critical analysis of urea transporter B inhibitors: molecular fingerprints, pharmacophore features for the development of next-generation diuretics

2022

Predictive Comparative QSAR Modeling of 4-Pyridones as Potent Antimalarials

2010

Cholesteryl ester transfer protein inhibitors in coronary heart disease: Validated comparative QSAR modeling of N, N-disubstituted trifluoro-3-amino-2-propanols

Computers in Biology and Medicine · 1970 · journal article

Chemoimmunotherapeutic approach to prolonged survival time in combination with immunization and glutamic acid derivatives with antitumor activity in tumor-bearing mice

Biological and Pharmaceutical Bulletin · 1970 · journal article

Structural finding of R/S-3,4-dihydro-2,2-dimethyl-6-halo-4-(substituted phenylaminocarbonylamino)-2H-1-benzopyrans as selective pancreatic β-cells K<inf>ATP-pβ</inf> channel openers

Canadian Journal of Chemistry · 1970 · journal article

Quantitative structure-activity relationship study on some azidopyridinyl neonicotinoid insecticides for their selective affinity towards the Drosophila nicotinic receptor over mammalian α<inf>4</inf>β<inf>2</inf> receptor using electrotopological state atom index

Drug Design and Discovery · 1970 · journal article

Photodynamic activity attained through the ruptured π-conjugation of pyridyl groups with a porphyrin macrocycle: Synthesis and the photophysical and photobiological evaluation of 5-mono-(4-nitrophenyl)-10,15,20-tris-[4-(phenoxymethyl)pyridine]-porphyrin and its Zn(ii) complex

Photochemical and Photobiological Sciences · 1970 · journal article

Exploring different classification-dependent QSAR modelling strategies for HDAC3 inhibitors in search of meaningful structural contributors

2024

Exploration of Fingerprints and Data Mining-based Prediction of Some Bioactive Compounds from Allium sativum as Histone Deacetylase 9 (HDAC9) Inhibitors

2024

Identification of structural fingerprints among natural inhibitors of HDAC1 to accelerate nature-inspired drug discovery in cancer epigenetics

2023

Host P2X7R-p38MAPK axis mediated intra-macrophage leishmanicidal activity of Spergulin-A

2022

QSAR for analogs of 1,5-N,N'-disubstituted-2-(substituted benzenesulphonyl) glutamamides as antitumor agents

2007

Pharmacophore Mapping of Tricyclic Isoxazoles for Their Affinity Towards Alpha-2 Adrenoreceptors #

2006

Unveiling structural components of dibenzofuran-based MMP-12 inhibitors: a comparative classification-dependent analysis with molecular docking-based virtual screening and molecular dynamics simulation

2025

Chrysin-functionalized gold nanoparticles and paclitaxel exhibit synergistic impact on lung cancer cell lines via regulating the AKT/PPAR-ϒ/β-catenin pathway

2024

Exploring crucial structural attributes of quinolinyl methoxyphenyl sulphonyl-based hydroxamate derivatives as ADAM17 inhibitors through classification-dependent molecular modelling approaches

2024

Quasi-SMILES as a Tool for Peptide QSAR Modelling

2023

Dissecting the Drug Development Strategies Against SARS-CoV-2 Through Diverse Computational Modeling Techniques

2020

Evaluation of the antipyretic potential of methanol extract of the leaves of Abies spectabilis (D. Don) Spach.

2007

Microdontic maxillary lateral incisor: case report.

1992

A fragment-based exploration of diverse MMP-9 inhibitors through classification-dependent structural assessment

2023

HDAC9 as a Privileged Target: Reviewing its Role in Different Diseasesand Structure-activity Relationships (SARs) of its Inhibitors

2023

Therapies of Hematological Malignancies: An Overview of the Potential Targets and Their Inhibitors

2021

Structural findings of pyrazolo[1,5- a ]pyrimidine compounds for their Pim-1/2 kinase inhibition as potential anticancer agents

2017

Nitric Oxide Synthase (NOS) Inhibitors in Cancer Angiogenesis

2015

Search for Structural Requirements of 2-Phenylimidazo(1,2-. ) pyridineacetamide Analogs to Improve Affinity and Selectivity towards Central and/or Peripheral Benzodiazepine Receptors

2007

QSAR Study on Some Dihydrofolate Reductase Inhibitors

2003

Nitrogen-containing heterocycles as important scaffold for selective and potent HDAC8 inhibition: a step towards effective, non-toxic and selective HDAC8 inhibitor discovery

2024

2D-QSAR Studies

2023

3D-QSAR Studies

2023

In-house glutamine based compound loaded poly-(D-L-lactide-coglycolide) nanoparticles as a possible candidate for the management of chronic myeloid leukemia

2023

Exploring molecular fingerprints of different drugs having bile interaction: a stepping stone towards better drug delivery

2023

In Silico Discovery of Class IIb HDAC Inhibitors: The State of Art

2023

Predictive Quantitative Structure Toxicity Relationship Study on Avian Toxicity of Some Diverse Agrochemical Pesticides by Monte Carlo Method

2016

Axially-symmetric Neutron stars: Implication of rapid rotation

2009

Search for Potential Anticancer Agents: Evaluation of Anticancer Activity of Carcinosin, Apis and Thuja

2008

1,5-N,N'-Disubstituted-2-(Substituted Benzenesulphonyl)- Glutamamide Analogues as Anticancer Agents. Part 3. † Synthesis, Biological Screening and QSAR Study #

2005

Potential energy surfaces forN =Z,20Ne-112Ba nuclei

2004

Development of Indomethacin- and Ibuprofen-loaded Polymethylmethacrylate Microparticles

1996

Arylcarboxamide Derivatives as Promising HDAC8 Inhibitors: An Overview in Light of Structure-activity Relationship and Binding Mode of Interaction Analysis

2024

Modeling Inhibitors of Gelatinases

2023

Other Modeling Approaches

2023

Establishing connection between neutron star properties and nuclear matter parameters through a comprehensive multivariate analysis

2023

Exploring Structural Requirements of Diarylurea Derivatives as VEGFR-2 Inhibitors Through Comparative QSAR Modeling Study

2020

First Report on the Validated Classification-Based Chemometric Modeling of Human Rhinovirus 3C Protease (HRV 3Cpro) Inhibitors

2018

Application of Computation in the Biosynthesis of Phytochemicals

2018

Epstein–Barr Virus and Treatment of Its Infection

2014

QSAR Study on Some Antirhino/Enteroviral Vinylacetylene Benzimidazoles

2003

QSAR Study on Some Substituted Glutamine Analogs as Anticancer Agents

2003

Effect of Λ<inf>v</inf> coupling on liquid gas phase transition in warm asymmetric nuclear matter

Nuclear Physics A · 1970 · journal article

Integrin antagonists: A special emphasis on structural requirements of n-benzoyl-l-biphenylalanines as α<inf>4</inf>β<inf>7</inf> and α<inf>4</inf>β<inf>1</inf> antagonists

Current Signal Transduction Therapy · 1970 · journal article

Possible anticancer agents: synthesis, pharmacological activity, and molecular modeling studies on some 5-N -Substituted-2-N-(substituted benzenesulphonyl)-L(+)Glutamines

Medicinal Chemistry Research · 1970 · journal article

Ligand- and structure- based drug design of non- steroidal aromatase inhibitors (NSAIs) in breast cancer

Oncology: Breakthroughs in Research and Practice · 1970 · book

Modeling Inhibitors of Membrane-Type MMPs

2023

Conclusion and Future Perspectives

2023

Modeling Inhibitors of Other MMPs

2023

Modeling Inhibitors of Collagenases

2023

Membrane-Type MMPs and Their Inhibitors

2023

Other MMPs and Their Inhibitors

2023

Collagenases and Their Inhibitors

2023

Stromelysins and Their Inhibitors

2023

Gelatinases and Their Inhibitors

2023

Modeling Inhibitors of Stromelysins

2023

Matrilysin and Their Inhibitors

2023

Modeling Inhibitors of Matrilysin

2023

Exploring Structural Requirements of HDAC10 Inhibitors Through Comparative Machine Learning Approaches

2023

Host P2X &lt;sub&gt;7&lt;/sub&gt;R-P &lt;sub&gt;38&lt;/sub&gt;MAPK Axis Mediated Intra-Macrophage Leishmanicidal Activity of Spergulin-A

2022

Apoptosis Inducing Activity of Diospyros melanoxylon Bark Extract on Molt-3 Cell Line via Activation of Mitochondrial Membrane Caspase Cascade and Cell Cycle Arrest with its Antioxidant Potential

2021

Synthesis, biological evaluation, and enzyme assay of some 5-N-substituted-2-N- (arylsulphonyl)-L(+)glutamines as potential anticancer agents

2020

Innovation Strategies to Cope Up with Globalization: How to Market Digital Nomads

2020

A Comparative Multi-QSAR Modelling and Molecular Docking Studies of Some Arylsulfonamide-Based ADAM17 Inhibitors as Anticancer Agents

2020

Discriminations of Actives from Inactives HDAC8 Inhibitors: Molecular Modeling Study to Explore Essential Molecular Fingerprints

2020

Exploring the Structural Aspects of Ureido Amino Acid-Based APN Inhibitors through Validated Comparative Regression and Classification Based Molecular Modeling Studies

2020

Contributors

2020

Spergulin-A strives intra-macrophage leishmanicidal activity by regulating the host P2X ₇ R-P ₃₈ MAPK axis

2019

Impact of Magnetic field on neutron star properties

2018

Contributors

2018

Supplementary material : Homoisoflavonoids as potential antiangiogenic agents for retinal neovascularization

2017

Iconography : Homoisoflavonoids as potential antiangiogenic agents for retinal neovascularization

2017

Contributors

2017

Development of Nitric Oxide Synthase (NOS) Inhibitors for Cancer Angiogenesis

2015

Properties of Rotating Neutron Star

2015

At a More Integrative Level It Examines and Index the Organic Pathways and Organizations that are a Significant Piece of Frameworks Science

2015

SP HSP-Exploration of structural and physicochemical requirements and search of virtual hits of HSP90 inhibitors as potential anticancer agents

2014

The rotating frequency and GW strain amplitude from Nuclear Models

2014

C onstraints on nuclear m atter param eters ofan Eective C hiralM odel

2013

Impact of a light stabilized radion in supernovae cooling

2012

POSSIBLE ANTINEOPLASTIC AGENTS, PART XVI: SYNTHESIS, IN VIVO ANTITUMOR AND INVITRO ANTIANGIOGENIC STUDY OF FEW GLUTAMIC ACID ANALOGS

2011

`$f_0 (600)$' and chiral dynamics

2009

From nuclear matter to Neutron Stars

2009

Calibration of nuclear matter parameters in an eective chiral model

2009

Search for Potential Anticancer Agents

2008

Effect of Hyperons on Nuclear Equation of State and Neutron Star Structure

2008

The island of deformation and shape co-existence in neutron-deficient nuclei of the Pb region using relativistic mean field model

2004

Role of BCS-type pairing in light deformed nuclei: A relativistic mean field approach

2003

ChemInform Abstract: POSSIBLE ANTINEOPLASTIC AGENTS: PART VIII ‐ SYNTHESIS AND ANTINEOPLASTIC ACTIVITY OF 5‐N‐SUBSTITUTED 3‐P‐SUBSTITUTED‐PHENYLGLUTARAMIC ACIDS AND 5‐N‐SUBSTITUTED 2‐BENZENESULFONYL‐3‐PHENYL‐L‐GLUTAMINES

1984

Towards the development of anticancer drugs from andrographolide: Semisynthesis, bioevaluation, QSAR analysis and pharmacokinetic studies

Current Topics in Medicinal Chemistry · 1970 · journal article

A new ellagic acid glycoside and DNA topoisomerase IB inhibitory activity of saponins from Putranjiva roxburghii

Natural Product Communications · 1970 · journal article

Epstein-barr virus and treatment of its infection

Cancer-Causing Viruses and their Inhibitors · 1970 · book chapter

Massive neutron stars and their implications

Pramana - Journal of Physics · 1970 · journal article

Tsallis statistics and the role of a stabilized radion in the supernovae SN1987A cooling

International Journal of Modern Physics A · 1970 · journal article

Predictive comparative QSAR modeling of 4-pyridones as potent antimalarials

Internet Electronic Journal of Molecular Design · 1970 · journal article

QSAR for analogs of 1,5-N,N'-disubstituted-2-(substituted benzenesulphonyl) glutamamides as antitumor agents

Internet Electronic Journal of Molecular Design · 1970 · journal article

QSAR study on coumarins as antimeningoencephalitic agents

Internet Electronic Journal of Molecular Design · 1970 · journal article

Possible antineoplastic agents, part XVI: Synthesis, In Vivo Antitumor and Invitro antiangiogenic study of few glutamic acid analogs

International Journal of Pharmaceutical Sciences Review and Research · 1970 · journal article

Predictive comparative QSAR modeling of 4-Pyridones as potent antimalarials

Internet Electronic Journal of Molecular Design · 1970 · journal article

QSAR study on coumarins as antimeningoencephalitic agents

Internet Electronic Journal of Molecular Design · 1970 · journal article

QSAR study on some orally active uracil derivatives as human gonadotropin-releasing-hormone receptor antagonists

Internet Electronic Journal of Molecular Design · 1970 · journal article

Antitumor activity and antioxidant role of Ichnocarpus frutescens against Ehrlich ascites carcinoma in Swiss albino mice

Natural Product Sciences · 1970 · journal article

Evaluation of the antipyretic potential of methanol extract of the leaves of Abies spectabilis (D. Don) Spach

Indian Journal of Natural Products and Resources · 1970 · journal article

QSAR for analogs of 1,5-N,N′-disubstituted-2-(substituted benzenesulphonyl) glutamamides as antitumor agents

Internet Electronic Journal of Molecular Design · 1970 · journal article

Search for structural requirements of 2-phenylimidazo[1,2-α] pyridineacetamide analogs to improve affinity and selectivity towards central and/or peripheral benzodiazepine receptors

Internet Electronic Journal of Molecular Design · 1970 · journal article

QSAR study on some synthesized and biologically evaluated glutamine analogs as possible anticancer agents

Indian Journal of Chemistry - Section A Inorganic, Physical, Theoretical and Analytical Chemistry · 1970 · journal article

Potential energy surfaces for N = Z, ²⁰Ne-¹¹²Ba nuclei

Pramana - Journal of Physics · 1970 · journal article

Shape change in HF, W and Os-isotopes: A non-relativistic Hartree-Fock versus relativistic Hartree approximation

Pramana - Journal of Physics · 1970 · journal article

A relativistic mean-field study of magic numbers in light nuclei from neutron to proton drip-lines

Pramana - Journal of Physics · 1970 · journal article

Enhanced regression of tumors in mice with combined chemotherapy and immunotherapy

Indian Journal of Pharmacology · 1970 · journal article

Syntheses, biological evaluation and QSAR study on antitumor activity of 1,5-N,N′-disubstituted-2-(substituted benzenesulphonyl) glutamamides

Bioorganic and Medicinal Chemistry · 1970 · journal article

Quantitative structure activity relationship (QSAR) studies of some substituted benzenesulphonyl glutamines as tumour suppressors.

Indian Journal of Biochemistry and Biophysics · 1970 · journal article

Development of indomethacin- and ibuprofen-loaded polymethylmethacrylate microparticles

Pharmaceutical Sciences · 1970 · journal article

Possible antineoplastic agents: Part XIII. Synthesis, biological evaluation and QSAR studies of some 1-(substituted benzenesulphonyl)-5-oxopyrrolldlne-2-carboxylic acid derivatives

Anti-Cancer Drug Design · 1970 · journal article

4-(4'-substituted benzoyl)aminobenzenesulphonyl-L(+)-glutamic acids and 5-N-substituted-2-[4'-(4''-substituted benzoyl)aminobenzenesulphonyl]-L-glutamines as potential antineoplastic agents: Synthesis, biological evaluation and quantitative structure-activity relationship studies

Indian Journal of Chemistry - Section B Organic Chemistry Including Medicinal Chemistry · 1970 · journal article

Possible antineoplastic agents X: Synthesis, antineoplastic activity and QSAR study of some 5-n-substituted-2-(chlorosubstituted benzenesulphonyl)-L-glutamines and 5-N-alkyl-2-(2',5'-dichlorobenzenesulphonyl)-L-glutamines

Indian Journal of Pharmaceutical Sciences · 1970 · journal article

Possible antineoplastic agents IX: Synthesis, antineoplastic activity and quantitative structure activity relationship of 5-N-substituted-2-(chlorosubstituted benzenesulphonyl)-L-glutamines

Indian Journal of Pharmaceutical Sciences · 1970 · journal article

Discriminations of active from inactive HDAC8 inhibitors Part II: Bayesian classification study to find molecular fingerprints

SAR and QSAR in Environmental Research · 1970 · journal article

Synthesis, biological evaluation, and enzyme assay of some 5-N-substituted-2-N-(arylsulphonyl)-L(+)glutamines as potential anticancer agents

Journal of the Indian Chemical Society · 1970 · journal article

Deconfinement of nonstrange hadronic matter with nucleons and Δ baryons to quark matter in neutron stars

International Journal of Modern Physics D · 1970 · journal article

Effects of hadron-quark phase transition on properties of neutron stars

Journal of Physics G: Nuclear and Particle Physics · 1970 · journal article

Properties of Neutron stars with hyperon cores in parametrized hydrostatic conditions

International Journal of Modern Physics E · 1970 · journal article

Structural findings of pyrazolo[1,5-a]pyrimidine compounds for their Pim-1/2 kinase inhibition as potential anticancer agents

Indian Journal of Biochemistry and Biophysics · 1970 · journal article

Nitric oxide synthase (NOS) inhibitors in cancer angiogenesis

Current Enzyme Inhibition · 1970 · journal article

Anthocephaline, a New Indole Alkaloid and Cadambine, a Potent Inhibitor of DNA Topoisomerase IB of Leishmania donovani (LdTOP1LS), Isolated from Anthocephalus cadamba

Natural Product Communications · 1970 · journal article